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本品为α-受体阻断药,通过阻断α-受体和间接激动β-受体,迅速使周围血管扩张,可显著降低外周血管阻力,增加周围血容量,改善微循环。本品对心脏有兴奋作用,使心肌收缩力增加、心率加快、心输出量增加。临床主要用于**肺充血或肺水肿的急性心力衰竭、血管痉挛性疾病、手足发绀症、感性中**休克及嗜铬细胞瘤的诊断试验等。亦用于室性早搏。
Adrenergic blocking agent. An antihypertensive. Used for the treatment of pheochromocytoma
甲磺酸酚妥拉明Phentolamine MesylateCAS号:65-28-1
甲磺酸酚妥拉明Phentolamine Mesylate分子式: C18H23N3O4S
甲磺酸酚妥拉明Phentolamine Mesylate英文名称: PHENTOLAMINE MESYLATE
甲磺酸酚妥拉明Phentolamine Mesylate英文同义词: VASOMAX; m-(n-(2-imidazolin-2-ylmethyl)-p-toluidino)-; phenomonomethanesulfonate(sal; phentolaminemethanesulphonate; phentolamine methanesulfonate; Phentolamine methanesulfonate salt; phentolamine mesilate; 3-[(4,5-dihydro-1H-imidazol-2-ylmethyl)(4-methylphenyl)amino]phenol methanesulfonate (1:1)
甲磺酸酚妥拉明Phentolamine MesylateEINECS号: 200-604-6
甲磺酸酚妥拉明Phentolamine Mesylate分子量: 377.4579
甲磺酸酚妥拉明Phentolamine Mesylate熔点: 180-182℃
甲磺酸酚妥拉明Phentolamine Mesylate沸点: 551°C at 760 mmHg
甲磺酸酚妥拉明Phentolamine Mesylate密度: 9.48E-13mmHg at 25°C
甲磺酸酚妥拉明Phentolamine Mesylate闪点: 287°C