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High quality FULVESTRANT,CAS No.129453-61-8,active pharmaceutical ingredient
Chemical Properties
Appearance:
white powder
Molecular Weight:
606.77
Density:
1.201 g/cm3
Boiling Point:
674.8 °C at 760 mmHg
Flash Point:
361.9 °C
Storage Temperature:
2-8°C
Refractive index:
1.521
Solubility:
In **, 9.53X10-6 mg/L at 25 deg C (est)
Biological Activity:
A high affinity estrogen receptor antagonist (IC 50 = 0.29 nM), devoid of any partial agonism both in vitro and in vivo . Also high affinity agonist at the membrane estrogen receptor GPR30.
Usage:
Antineoplastic (hormonal)
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